CYCLIZATION OF TRYPTAMINE ENAMINONES TO FUNCTIONALIZED TETRAHYDRO-BETA-CARBOLINES INDUCED BY [BIS(TRIFLUORCEACETOXY)IODO] BENZENE

Authors
PAPADOPOULOU D PAPOUTSIS I SPYROUDIS S VARVOGLIS A
Citation
D. Papadopoulou et al., CYCLIZATION OF TRYPTAMINE ENAMINONES TO FUNCTIONALIZED TETRAHYDRO-BETA-CARBOLINES INDUCED BY [BIS(TRIFLUORCEACETOXY)IODO] BENZENE, Tetrahedron letters, 39(18), 1998, pp. 2865-2866
Citations number
6
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
39
Issue
18
Year of publication
1998
Pages
2865 - 2866
Database
ISI
SICI code
0040-4039(1998)39:18<2865:COTETF>2.0.ZU;2-T
Abstract
The reaction of enamino carbonyl derivatives of tryptamine with [bis(t rifluoroacetoxy)iodo]benzene provides an easy route to ctionalised-N-t rifluoroacetylated-beta-carbolines. The reaction proceeds through Pict et-Spengler-type cyclisation, trifluoroacetylation and oxidation steps . (C) 1998 Elsevier Science Ltd. All rights reserved.