NEW ARYL HETEROARYL C-N BOND CROSS-COUPLING REACTIONS VIA ARYLBORONICACID CUPRIC ACETATE ARYLATION/

Authors
LAM PYS CLARK CG SAUBERN S ADAMS J WINTERS MP CHAN DMT COMBS A
Citation
Pys. Lam et al., NEW ARYL HETEROARYL C-N BOND CROSS-COUPLING REACTIONS VIA ARYLBORONICACID CUPRIC ACETATE ARYLATION/, Tetrahedron letters, 39(19), 1998, pp. 2941-2944
Citations number
15
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
39
Issue
19
Year of publication
1998
Pages
2941 - 2944
Database
ISI
SICI code
0040-4039(1998)39:19<2941:NAHCBC>2.0.ZU;2-0
Abstract
A new aryl/heteroaryl C-N bond cross-coupling reaction via the arylbor onic acid/cupric acetate arylation of N-H containing heteroarenes has been discovered. This new methodology is mild, proceeds at room temper ature exposed to air, and works for many heteroarenes and arylboronic acids providing good yields of N-arylated heteroarenes. (C) 1998 Elsev ier Science Ltd. All rights reserved.