Rs. Mali et Ap. Massey, SYNTHESIS OF NATURALLY-OCCURRING 5-ALLYL-2-ARYL-7-METHOXYBENZOFURAN AND 2-ARYL-5-(3-HYDROXYPROPYL)-7-METHOXYBENZOFURANS, Journal of chemical research. Synopses (Print), (5), 1998, pp. 230
A convenient and general procedure is described for the synthesis of 5
-allyl-2-aryl-7-methoxybenzofurans (8a-e) from 2-allyloxy-3-methoxyben
zaldehyde (3). The compounds 8a and 8b on hydroboration followed by ox
idation provide the naturally occurring benzofurans (1a and 1b).