M. Barbier et al., SYNTHESIS OF ISOBRASSILEXIN, A BIOLOGICALLY-ACTIVE ISOMER OF BRASSILEXIN, A CRUCIFERAE PHYTOALEXIN, Synthetic communications, 23(22), 1993, pp. 3109-3117
The synthesis of isobrassilexin 2,a hitherto non natural indoloisothia
zole is reported (two steps, 43% yield). This substance, an isomer of
brassilexin 1 has shown important biological properties in vitro.