Palladium catalyzed cross-coupling reaction of stereodefined cyclopropylboronic acids with N-heterocycl bromides

Authors
Ma, HR Wang, XH Deng, MZ
Citation
Hr. Ma et al., Palladium catalyzed cross-coupling reaction of stereodefined cyclopropylboronic acids with N-heterocycl bromides, SYN COMMUN, 29(14), 1999, pp. 2477-2485
Citations number
10
Categorie Soggetti
Organic Chemistry/Polymer Science
Journal title
SYNTHETIC COMMUNICATIONS
ISSN journal
00397911 → ACNP
Volume
29
Issue
14
Year of publication
1999
Pages
2477 - 2485
Database
ISI
SICI code
0039-7911(1999)29:14<2477:PCCROS>2.0.ZU;2-E
Abstract
The Suzuki-type cross-coupling reaction of stereodefined cyclopropylboronic acids with N-heterocycl bromides was investigated. In the appropriate cond itions the coupling reactions readily underwent to afford stereocontrolled cyclopropyl substituted N-heterocycles in moderate to good yields. The conf iguration of cycloplopylboronic acids retained during the reaction.