Synthesis of pyrrolidine or piperidine ring-fused azepino[5,4,3-cd]indole derivatives

Citation
Ys. Lee et al., Synthesis of pyrrolidine or piperidine ring-fused azepino[5,4,3-cd]indole derivatives, TETRAHEDR L, 40(30), 1999, pp. 5569-5572
Citations number
18
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
TETRAHEDRON LETTERS
ISSN journal
00404039 → ACNP
Volume
40
Issue
30
Year of publication
1999
Pages
5569 - 5572
Database
ISI
SICI code
0040-4039(19990723)40:30<5569:SOPOPR>2.0.ZU;2-C
Abstract
The synthesis of pyrrolidine or piperidine ring-fused 2-phenylazepino[5,4,3 -cd]indole derivatives (2) has been accomplished through the N-acyliminium ion cyclization of hydroxy- or alkoxylactams (5) derived from cyclic anhydr ides or chiral hydroxy acids. (C) 1999 Elsevier Science Ltd. All rights res erved.