A versatile new synthesis of 4-aryl- and heteroaryl[3,4-c]pyrrolocarbazoles by [4+2] cycloaddition followed by palladium catalysed cross coupling

Authors
McCort, G Duclos, O Cadilhac, C Guilpain, E
Citation
G. Mccort et al., A versatile new synthesis of 4-aryl- and heteroaryl[3,4-c]pyrrolocarbazoles by [4+2] cycloaddition followed by palladium catalysed cross coupling, TETRAHEDR L, 40(34), 1999, pp. 6211-6215
Citations number
13
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
TETRAHEDRON LETTERS
ISSN journal
00404039 → ACNP
Volume
40
Issue
34
Year of publication
1999
Pages
6211 - 6215
Database
ISI
SICI code
0040-4039(19990820)40:34<6211:AVNSO4>2.0.ZU;2-C
Abstract
4-Bromo- and 4-trifluorosulfonyloxypyrrolo[3,4-c]carbazoles were prepared i n five steps via a [4+2] cycloaddition and were used as key intermediates i n palladium-catalysed cross coupling reactions allowing the rapid generatio n of structurally diverse protein kinase C inhibitors. (C) 1999 Published b y Elsevier Science Ltd. All rights reserved.