The synthesis of aminoazole analogs of lysine and arginine: The Mitsunobu reaction with lysinol and argininol

Authors
Citation
Ho. Kim et M. Kahn, The synthesis of aminoazole analogs of lysine and arginine: The Mitsunobu reaction with lysinol and argininol, SYNLETT, (8), 1999, pp. 1239-1240
Citations number
6
Categorie Soggetti
Organic Chemistry/Polymer Science
Journal title
SYNLETT
ISSN journal
09365214 → ACNP
Issue
8
Year of publication
1999
Pages
1239 - 1240
Database
ISI
SICI code
0936-5214(199908):8<1239:TSOAAO>2.0.ZU;2-X
Abstract
The Mitsunobu reaction of aminooxazoles and thiazoles with lysinol and argi ninol is described. The aminooxazoles and thiazoles reacted with lysinol or argininol in the presence of triphenylphosphine and dialkyl azodicarboxyla te to provide the reduced peptidyl azoles in moderate to good yields.