Ho. Kim et M. Kahn, The synthesis of aminoazole analogs of lysine and arginine: The Mitsunobu reaction with lysinol and argininol, SYNLETT, (8), 1999, pp. 1239-1240
The Mitsunobu reaction of aminooxazoles and thiazoles with lysinol and argi
ninol is described. The aminooxazoles and thiazoles reacted with lysinol or
argininol in the presence of triphenylphosphine and dialkyl azodicarboxyla
te to provide the reduced peptidyl azoles in moderate to good yields.