A general inhibitor scaffold for serine proteases with a (chymo)trypsin-like fold: Solution-phase construction and evaluation of the first series of libraries of mechanism-based inhibitors
Rz. Kuang et al., A general inhibitor scaffold for serine proteases with a (chymo)trypsin-like fold: Solution-phase construction and evaluation of the first series of libraries of mechanism-based inhibitors, J AM CHEM S, 121(35), 1999, pp. 8128-8129