Citation
D. Passarella et al., Convenient synthesis of methyl indol-2-ylpropiolate, J CHEM S P1, (19), 1999, pp. 2669-2670
Citations number
26
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1
ISSN journal
0300922X
→ ACNP
Issue
19
Year of publication
1999
Pages
2669 - 2670
Database
ISI
SICI code
0300-922X(1999):19<2669:CSOMI>2.0.ZU;2-Q
Abstract
Methyl indol-2-ylpropiolate 1 is synthesized by using a catalyst system of
PPh3-CuI in the presence of K2CO3 as base. The procedure appears convenient
if compared with Pd-catalyzed cross-coupling reactions. The interest is in
creased by the use of an alk-1-yne containing an electron-withdrawing group
.