A convenient method for the synthesis of six-membered heterocyclic enaminones

Authors
Puebla, P Honores, Z Medarde, M Caballero, E San Feliciano, A Moran, L
Citation
P. Puebla et al., A convenient method for the synthesis of six-membered heterocyclic enaminones, J HETERO CH, 36(4), 1999, pp. 1097-1099
Citations number
8
Categorie Soggetti
Organic Chemistry/Polymer Science
Journal title
JOURNAL OF HETEROCYCLIC CHEMISTRY
ISSN journal
0022152X → ACNP
Volume
36
Issue
4
Year of publication
1999
Pages
1097 - 1099
Database
ISI
SICI code
0022-152X(199907/08)36:4<1097:ACMFTS>2.0.ZU;2-R
Abstract
Enaminones are widely employed in the synthesis of heterocycles, however he terocyclic enaminones and their use in the synthesis of more complex system s have been less studied. The reaction between 4-chloroacetylacetate and al iphatic or aromatic 1,2-aminoalcohols, 1,2-aminothiols or 1,2-diamines, yie lds in one pot a six-membered 1,4-heterocyclic system containing the enamin one moiety.