The chemistry of indoles Part 94 - A novel methodology for preparing 5-chloro- and 5-bromotryptamines and tryptophans, and its application to the synthesis of (+/-)-bromochelonin B

Authors
Hasegawa, M Yamada, K Nagahama, Y Somei, M
Citation
M. Hasegawa et al., The chemistry of indoles Part 94 - A novel methodology for preparing 5-chloro- and 5-bromotryptamines and tryptophans, and its application to the synthesis of (+/-)-bromochelonin B, HETEROCYCLE, 51(12), 1999, pp. 2815-2821
Citations number
13
Categorie Soggetti
Organic Chemistry/Polymer Science
Journal title
HETEROCYCLES
ISSN journal
03855414 → ACNP
Volume
51
Issue
12
Year of publication
1999
Pages
2815 - 2821
Database
ISI
SICI code
0385-5414(199912)51:12<2815:TCOIP9>2.0.ZU;2-R
Abstract
A novel methodology for introducing chlorine or bromine into the 5-position of tryptamines was found through 1-hydroxytryptamines. The chemistry was a pplied to the syntheses of(+/-)5-chloro-, -5-bromotryptophan derivatives, a nd (+/-)-bromochelonin B.