The Mukaiyama-Michael reaction of N-acyl-2,3-dihydro-4-pyridones: Regio- and stereoselective synthesis of cis-2,6-disubstituted 1,2,5,6-tetrahydropyridines
Jt. Kuethe et Dl. Comins, The Mukaiyama-Michael reaction of N-acyl-2,3-dihydro-4-pyridones: Regio- and stereoselective synthesis of cis-2,6-disubstituted 1,2,5,6-tetrahydropyridines, ORG LETT, 1(7), 1999, pp. 1031-1033
[GRAPHICS]
A convenient regio- and stereoselective preparation of 1,2,5,6-tetrahydropy
ridines of the type 1 has been developed, starting from readily available N
-acyl-2,2-dihydro-4-pyridones 2.