Palladium-catalyzed functionalization of 5-and 7-azaindoles

Authors
Chi, SM Choi, JK Yum, EK Chi, DY
Citation
Sm. Chi et al., Palladium-catalyzed functionalization of 5-and 7-azaindoles, TETRAHEDR L, 41(6), 2000, pp. 919-922
Citations number
26
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
TETRAHEDRON LETTERS
ISSN journal
00404039 → ACNP
Volume
41
Issue
6
Year of publication
2000
Pages
919 - 922
Database
ISI
SICI code
0040-4039(20000205)41:6<919:PFO57>2.0.ZU;2-U
Abstract
Palladium-catalyzed functionalization at the 2-position of various 5- and 7 -azaindoles was performed by Suzuki, Heck, and Stille reactions. The 2-subs tituted azaindoles were obtained with 5% Pd(OAc)(2), LiCl, and KOAc in DMF at 110 degrees C with moderate to high yields. (C) 2000 Elsevier Science Lt d. All rights reserved.