Pj. Bhuyan et al., Studies on uracils: an efficient method for the synthesis of novel 1-allyl-6-(1 ',2 ',3 '-triazolyl) analogues of HEPT, J CHEM S P1, (21), 1999, pp. 3083-3084
An efficient synthetic method for preparing novel 1-allyl-6-(1',2',3'-triaz
olyl) analogues of HEPT, an anti-HIV reverse transcriptase inhibitor, is re
ported. The key step is based upon selective intermolecular cycloaddition o
f azide to acetylenes.