Rs. Garigipati et al., NOVEL FRAMEWORKS FOR TRIFLUOROMETHYL KETONE AND PHOSPHONATE TSA INHIBITORS OF TYPE-II PLA(2), Bioorganic & medicinal chemistry letters, 7(11), 1997, pp. 1421-1426
Design and synthesis of some TSA inhibitors on novel molecular framewo
rks is described. This TSA analog design culminates in the preparation
of the phosphonate 18. (C) 1997 Elsevier Science Ltd.