Traceless linking of indoles: General methodology and application to solidphase supported Mannich and Stille reactions

Citation
J. Kraxner et al., Traceless linking of indoles: General methodology and application to solidphase supported Mannich and Stille reactions, SYNLETT, (1), 2000, pp. 125-127
Citations number
23
Categorie Soggetti
Organic Chemistry/Polymer Science
Journal title
SYNLETT
ISSN journal
09365214 → ACNP
Issue
1
Year of publication
2000
Pages
125 - 127
Database
ISI
SICI code
0936-5214(200001):1<125:TLOIGM>2.0.ZU;2-J
Abstract
Transacetalization reaction of the diethoxymethyl (DEM) protected indoles 2 a,b,d,e with the polymer bound glycerol derivative 3 resulted in formation of the immobilized indoles 4a,b,d,e. Selective indole-functionalizations as well as quantitative and traceless cleavage could be demonstrated.