A practical synthesis of peptide mimetics via the solid-phase Petasis reaction

Authors
Klopfenstein, SR Chen, JJ Golebiowski, A Li, M Peng, SX Shao, X
Citation
Sr. Klopfenstein et al., A practical synthesis of peptide mimetics via the solid-phase Petasis reaction, TETRAHEDR L, 41(25), 2000, pp. 4835-4839
Citations number
26
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
TETRAHEDRON LETTERS
ISSN journal
00404039 → ACNP
Volume
41
Issue
25
Year of publication
2000
Pages
4835 - 4839
Database
ISI
SICI code
0040-4039(20000619)41:25<4835:APSOPM>2.0.ZU;2-B
Abstract
The boronic acid Mannich reaction (Petasis reaction) is demonstrated on a s olid support. Peptide mimetics are formed from N-alkylated amino acid resin esters, glyoxylic acid and boronic acids. (C) 2000 Elsevier Science Ltd. A ll rights reserved.