(N)UNDER-BAR-METHYL AS A BIOISOSTERE FOR THE OXYGEN LINK BETWEEN THE AROMATIC RINGS OF ARYLOXYPHENOXYPROPIONATE HERBICIDES

Authors
BIRD GJ CROSS LE FARQUHARSON GJ JENSEN WA LYDIATE J SERBAN A WARNER RB WATSON KG BARTON JED COLES C COLLINS DJ SLATER JW
Citation
Gj. Bird et al., (N)UNDER-BAR-METHYL AS A BIOISOSTERE FOR THE OXYGEN LINK BETWEEN THE AROMATIC RINGS OF ARYLOXYPHENOXYPROPIONATE HERBICIDES, Bioorganic & medicinal chemistry letters, 7(12), 1997, pp. 1489-1492
Citations number
10
Categorie Soggetti
Chemistry Inorganic & Nuclear","Chemistry Medicinal
Journal title
Bioorganic & medicinal chemistry letters → ACNP
ISSN journal
0960894X
Volume
7
Issue
12
Year of publication
1997
Pages
1489 - 1492
Database
ISI
SICI code
0960-894X(1997)7:12<1489:(AABFT>2.0.ZU;2-X
Abstract
The herbicidal activity of a set of (N) under bar,methyl arylaminophen oxypropionate esters 3 has been compared to the analogous aryloxypheno xypropionates 1. The usefulness of (N) under bar-methyl as a novel bio isostere for ether links is shown by the surprisingly high herbicidal activity of the 6-chloroquinazolin-2-yl- and -benzotriazin-3-yl-N-meth ylamino-phenoxypropionate esters 3h and 3i. (C) 1997 Elsevier Science Ltd.