Synthesis and systemic fungicidal activity of silicon-containing azole derivatives

Authors
Itoh, H Yoneda, R Tobitsuka, J Matsuhisa, T Kajino, H Ohta, H Hayashi, N Takahi, Y Tsuda, M Takeshiba, H
Citation
H. Itoh et al., Synthesis and systemic fungicidal activity of silicon-containing azole derivatives, CHEM PHARM, 48(8), 2000, pp. 1148-1153
Citations number
19
Categorie Soggetti
Chemistry & Analysis
Journal title
CHEMICAL & PHARMACEUTICAL BULLETIN
ISSN journal
00092363 → ACNP
Volume
48
Issue
8
Year of publication
2000
Pages
1148 - 1153
Database
ISI
SICI code
0009-2363(200008)48:8<1148:SASFAO>2.0.ZU;2-L
Abstract
A new series of azole derivatives containing silicon were synthesized and e valuated for fungicidal activity against rice sheath blight by submerged ap plication. Among them, 2-(4-fluorophenyl)-1-(1H-1,2,4-triazol-1-yl)-3-trime thylsilylpropan-2-ol (9a) exhibited satisfactory efficacy at 12.5 grams per 10 ares.