An activated phosphate for an efficient amide and peptide coupling reagent

Authors
Yasuhara, T Nagaoka, Y Tomioka, K
Citation
T. Yasuhara et al., An activated phosphate for an efficient amide and peptide coupling reagent, J CHEM S P1, (17), 2000, pp. 2901-2902
Citations number
35
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1
ISSN journal
14704358 → ACNP
Issue
17
Year of publication
2000
Pages
2901 - 2902
Database
ISI
SICI code
1470-4358(2000):17<2901:AAPFAE>2.0.ZU;2-P
Abstract
Activation of diethyl phosphate was realized by attaching trifluoromethanes ulfonanilide as an efficient leaving group and the phosphate 1 proved to be a promising amide and peptide coupling reagent.