Nn. Makhova et al., Effective synthesis of 1,2-di-, 1,2,3-tri-, 1,2,3,3-tetraalkyldiaziridinesand 1,5-diazabicyclo[3.1.0]hexanes, MENDELEEV C, (5), 2000, pp. 182-184
A versatile single-step procedure was proposed for the synthesis of the tit
le compounds by the interaction of equimolar amounts of aliphatic carbonyl
compounds, primary aliphatic amines and N-chloroalkylamines in an aprotic o
rganic solvent in the presence of potassium carbonate.