A concise preparation of yuehchukene and its analogues

Citation
M. Ishikura et al., A concise preparation of yuehchukene and its analogues, HETEROCYCLE, 53(10), 2000, pp. 2201
Citations number
42
Categorie Soggetti
Organic Chemistry/Polymer Science
Journal title
HETEROCYCLES
ISSN journal
03855414 → ACNP
Volume
53
Issue
10
Year of publication
2000
Database
ISI
SICI code
0385-5414(20001001)53:10<2201:ACPOYA>2.0.ZU;2-N
Abstract
The palladium catalyzed carbonylative cross-coupling reaction of indolylbor ates (2) with vinyl triflates (3) afforded indol-2-yl ketones (4), which we re subsequently converted to hexahydroindeno[2,1-b]indoles (5) with the aid of an acid. This protocol was well adapted for the total synthesis of yueh chukene.