An efficient synthesis of N-benzyl-3-sulfonyl glutarimides. Formal synthesis of the aromatase inhibitor AG-1

Authors
Chang, MY Chang, BR Tai, HM Chang, NC
Citation
My. Chang et al., An efficient synthesis of N-benzyl-3-sulfonyl glutarimides. Formal synthesis of the aromatase inhibitor AG-1, TETRAHEDR L, 41(52), 2000, pp. 10273-10276
Citations number
17
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
TETRAHEDRON LETTERS
ISSN journal
00404039 → ACNP
Volume
41
Issue
52
Year of publication
2000
Pages
10273 - 10276
Database
ISI
SICI code
0040-4039(200012)41:52<10273:AESONG>2.0.ZU;2-U
Abstract
A formal [3+3] cycloaddition strategy to substituted glutarimides was studi ed. N-Benzyl alpha -sulfonyl-acetamides and various alpha,beta -unsaturated esters were used as starting materials. (C) 2000 Elsevier Science Ltd. All rights reserved.