Access to pyrralo- and pyrido[1,2-a]indole derivatives by intramolecular nitrone cycloadditions. Effect of steric factors on the regioselective product formation

Citation
Em. Beccalli et al., Access to pyrralo- and pyrido[1,2-a]indole derivatives by intramolecular nitrone cycloadditions. Effect of steric factors on the regioselective product formation, J ORG CHEM, 65(26), 2000, pp. 8924-8932
Citations number
24
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
JOURNAL OF ORGANIC CHEMISTRY
ISSN journal
00223263 → ACNP
Volume
65
Issue
26
Year of publication
2000
Pages
8924 - 8932
Database
ISI
SICI code
0022-3263(200012)65:26<8924:ATPAPD>2.0.ZU;2-8
Abstract
On starting from N-allyl-substituted 2-indolecarbaldehydes and exploiting t he intramolecular nitrone cycloaddition methodology, we synthesized a numbe r of the title fused-ring indole derivatives in racemic as well as enantiop ure form.