Synthesis and cyclization of carboxylsulfamides derived from amines and alpha-hydroxyesters - Evaluation of bacteriostatic activity

Authors
Berredjema, M Regainia, Z Djahoudia, A Aoufa, NE Dewynter, G Monterob, JL
Citation
M. Berredjema et al., Synthesis and cyclization of carboxylsulfamides derived from amines and alpha-hydroxyesters - Evaluation of bacteriostatic activity, PHOSPHOR SU, 165, 2000, pp. 249-264
Citations number
18
Categorie Soggetti
Inorganic & Nuclear Chemistry
Journal title
PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS
ISSN journal
10426507 → ACNP
Volume
165
Year of publication
2000
Pages
249 - 264
Database
ISI
SICI code
1042-6507(2000)165:<249:SACOCD>2.0.ZU;2-2
Abstract
The synthesis of carboxylsulfamides was carried out starting from chlorosul fonyl isocyanate, primary amines and alpha -hydroxyesters. After reduction, the carboxylsulfamides were cyclised under Mitsunobu conditions giving N-s ulfamoyloxazolidinones in good yields.