M. Billet et al., Syn diastereoselectivity in the synthesis of homoallylamine using crotylsilane in the three-component reaction, TETRAHEDR L, 42(4), 2001, pp. 631-634
Crotylsilane was used in a three-component reaction for the synthesis of ho
moallylamines from aldehydes. A moderate to good syn/anti 5/1 diastereosele
ctivity was observed. The obtained homoallylamines were transformed into py
rrolidines or piperidines. (C) 2001 Elsevier Science Ltd. All rights reserv
ed.