A novel procedure for the synthesis of aziridines: application of Simmons-Smith reagents to aziridination

Authors
Aggarwal, VK Stenson, RA Jones, RVH Fieldhouse, R Blacker, J
Citation
Vk. Aggarwal et al., A novel procedure for the synthesis of aziridines: application of Simmons-Smith reagents to aziridination, TETRAHEDR L, 42(8), 2001, pp. 1587-1589
Citations number
29
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
TETRAHEDRON LETTERS
ISSN journal
00404039 → ACNP
Volume
42
Issue
8
Year of publication
2001
Pages
1587 - 1589
Database
ISI
SICI code
0040-4039(20010219)42:8<1587:ANPFTS>2.0.ZU;2-V
Abstract
The reaction of Simmons-Smith carbenoids with imines in the presence of sul fides provides N-(p-toluenesulfonyl)- and N-[(1,1,1-trimethylsilyl)ethyl]su lfonyl-substituted aziridines in high yield. (C) 2001 Elsevier Science Ltd. All rights reserved.