Efficient one-step synthesis of 3-amino-6-arylpyridazines

Authors
Guery, S Parrot, I Rival, Y Wermuth, CG
Citation
S. Guery et al., Efficient one-step synthesis of 3-amino-6-arylpyridazines, TETRAHEDR L, 42(11), 2001, pp. 2115-2117
Citations number
16
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
TETRAHEDRON LETTERS
ISSN journal
00404039 → ACNP
Volume
42
Issue
11
Year of publication
2001
Pages
2115 - 2117
Database
ISI
SICI code
0040-4039(20010311)42:11<2115:EOSO3>2.0.ZU;2-7
Abstract
Starting from the commercially available 3-amino-6-chloropyridazine, 3-amin o-6-arylpyridazines were prepared in good yields by means of a Suzuki cross -coupling reaction avoiding the somewhat lengthy four-step classic synthesi s. (C) 2001 Elsevier Science Ltd. All rights reserved.