A practical one-pot synthesis of 2,3-disubstituted indoles from unactivated anilines

Authors
Tokunaga, M Ota, M Haga, MA Wakatsuki, Y
Citation
M. Tokunaga et al., A practical one-pot synthesis of 2,3-disubstituted indoles from unactivated anilines, TETRAHEDR L, 42(23), 2001, pp. 3865-3868
Citations number
25
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
TETRAHEDRON LETTERS
ISSN journal
00404039 → ACNP
Volume
42
Issue
23
Year of publication
2001
Pages
3865 - 3868
Database
ISI
SICI code
0040-4039(20010604)42:23<3865:APOSO2>2.0.ZU;2-2
Abstract
2-Substituted-3-methyl indoles are synthesized with good regioselectivity f rom readily available substrates and catalysts, i.e. the reaction of anilin es with propargyl alcohols in the presence of 0.36-1 mol% Ru-3(CO)(12). (C) 2001 Elsevier Science Ltd. All rights reserved.