Synthesis of novel isothiazolo[4,3-b]pyridine and isothiazolo[4,3-b]quinoline derivatives

Authors
Wojciechowski, K Kosinski, S
Citation
K. Wojciechowski et S. Kosinski, Synthesis of novel isothiazolo[4,3-b]pyridine and isothiazolo[4,3-b]quinoline derivatives, TETRAHEDRON, 57(23), 2001, pp. 5009-5014
Citations number
14
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
TETRAHEDRON
ISSN journal
00404020 → ACNP
Volume
57
Issue
23
Year of publication
2001
Pages
5009 - 5014
Database
ISI
SICI code
0040-4020(20010604)57:23<5009:SONIAI>2.0.ZU;2-4
Abstract
The efficient synthesis of isothiazolo[4,3-b]pyridines and isothiazolo[4,3- b]quinolines via intramolecular vicarious nucleophilic substitution of hydr ogen in N-oxides and quaternary salts of chloromethanesulfonamides derived from 3-aminopyridine and 3-aminoquinoline is described. (C) 2001 Elsevier S cience Ltd. All rights reserved.