Selective palladium-catalyzed aminations on dichloropyridines

Authors
Jonckers, THM Maes, BUW Lemiere, GLF Dommisse, R
Citation
Thm. Jonckers et al., Selective palladium-catalyzed aminations on dichloropyridines, TETRAHEDRON, 57(32), 2001, pp. 7027-7034
Citations number
48
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
TETRAHEDRON
ISSN journal
00404020 → ACNP
Volume
57
Issue
32
Year of publication
2001
Pages
7027 - 7034
Database
ISI
SICI code
0040-4020(20010806)57:32<7027:SPAOD>2.0.ZU;2-E
Abstract
Palladium-catalyzed amination proved to be a valuable strategy for the sele ctive introduction of aromatic and heteroaromatic amines, including aminopy ridines and aminodiazines, on dichloropyridines. The use of mild amination conditions resulted in maximum selectivity and excellent base sensitive fun ctional group tolerance. (C) 2001 Elsevier Science Ltd. All rights reserved .