Jj. Turner et al., Synthesis of novel amino acid carbohydrate hybrids via Mitsunobu glycosylation of nitro benzenesulfonamides, TETRAHEDR L, 42(33), 2001, pp. 5763-5767
Amino acid derived 2-nitrobenzenesulfonamides were successfully condensed u
nder Mitsunobu conditions with the primary alcohol of various saccharide an
d nucleoside derivatives to furnish the fully protected hybrids in excellen
t yield. One such hybrid was incorporated into a short peptide sequence in
good overall yield. (C) 2001 Elsevier Science Ltd. All rights reserved.