Synthesis of 3-chloroanthranilates from alpha,gamma,gamma-trichloro-beta-iminoesters

Authors
Stevens, CV Kesteleyn, B Alonso, ER De Kimpe, N
Citation
Cv. Stevens et al., Synthesis of 3-chloroanthranilates from alpha,gamma,gamma-trichloro-beta-iminoesters, TETRAHEDRON, 57(36), 2001, pp. 7685-7692
Citations number
20
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
TETRAHEDRON
ISSN journal
00404020 → ACNP
Volume
57
Issue
36
Year of publication
2001
Pages
7685 - 7692
Database
ISI
SICI code
0040-4020(20010903)57:36<7685:SO3FA>2.0.ZU;2-Y
Abstract
3-Chloroanthranilates have been prepared by a short pathway involving dehyd rohalogenation of alpha,gamma,gamma -trichloro-beta -iminoesters, which wer e obtained by trihalogenation of the corresponding enaminoesters. This rout e opens the way to a number of previously unknown functionalised anthranila tes, which are potential starting materials for a variety of heterocyclic a nd biologically interesting compounds. (C) 2001 Elsevier Science Ltd. All r ights reserved.