3-Acyl-1,3-diaryltriazenes as neutral and selective acylating agents

Citation
B. Stefane et al., 3-Acyl-1,3-diaryltriazenes as neutral and selective acylating agents, TETRAHEDR L, 42(38), 2001, pp. 6659-6662
Citations number
20
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
TETRAHEDRON LETTERS
ISSN journal
00404039 → ACNP
Volume
42
Issue
38
Year of publication
2001
Pages
6659 - 6662
Database
ISI
SICI code
0040-4039(20010917)42:38<6659:3ANASA>2.0.ZU;2-1
Abstract
New 3-acyl-1,3-diaryltriazenes have been prepared and their reactions with amino compounds have been studied. Reactions proceed rapidly under mild con ditions to give the corresponding N-acyl products: Reagents enable chemosel ective acylation of aliphatic primary and secondary amines in the presence of other acylable functional groups. (C) 2001 Elsevier Science Ltd. All rig hts reserved.