Synthesis of Delta(1)-1,2-diazetines via a Diels-Alder cycloaddition approach

Authors
Breton, GW Shugart, JH Hughey, CA Perala, SM Hicks, AD
Citation
Gw. Breton et al., Synthesis of Delta(1)-1,2-diazetines via a Diels-Alder cycloaddition approach, ORG LETT, 3(20), 2001, pp. 3185-3187
Citations number
12
Categorie Soggetti
Organic Chemistry/Polymer Science
Journal title
ORGANIC LETTERS
ISSN journal
15237060 → ACNP
Volume
3
Issue
20
Year of publication
2001
Pages
3185 - 3187
Database
ISI
SICI code
1523-7060(20011004)3:20<3185:SODVAD>2.0.ZU;2-I
Abstract
GRAPHICS A novel method for the synthesis of Delta (1)-1,2-diazetines is presented. Diels-Alder cycloaddition of dienophile 4 with five dienes afforded cycload ducts in good to excellent yields. Four of the obtained cycloadducts were c onverted to the corresponding diazetines.