2-arylsulfinylmethyl oxazines: Chiral carbonyl equivalents

Citation
K. Singh et al., 2-arylsulfinylmethyl oxazines: Chiral carbonyl equivalents, HETEROCYCLE, 55(10), 2001, pp. 1937
Citations number
14
Categorie Soggetti
Organic Chemistry/Polymer Science
Journal title
HETEROCYCLES
ISSN journal
03855414 → ACNP
Volume
55
Issue
10
Year of publication
2001
Database
ISI
SICI code
0385-5414(20011001)55:10<1937:2OCCE>2.0.ZU;2-H
Abstract
A single pot acid catalysed condensation reaction of 2-arylsulfinylmethylox azinane - a chiral carbonyl equivalent (derived from the title oxazine by B H4- reduction) with tryptamine and tryptophan esters, furnishes tetrahydro- beta -carbolines and can be subsequently transformed into indole alkaloids.