X-ray crystal structure of a bisubstrate inhibitor bound to the enzyme catechol-O-methyltransferase: A dramatic effect of inhibitor preorganization on binding affinity

Authors
Lerner, C Ruf, A Gramlich, V Masjost, B Zurcher, G Jakob-Roetne, R Borroni, E Diederich, F
Citation
C. Lerner et al., X-ray crystal structure of a bisubstrate inhibitor bound to the enzyme catechol-O-methyltransferase: A dramatic effect of inhibitor preorganization on binding affinity, ANGEW CHEM, 40(21), 2001, pp. 4040
Citations number
19
Categorie Soggetti
Chemistry & Analysis",Chemistry
Journal title
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
ISSN journal
14337851 → ACNP
Volume
40
Issue
21
Year of publication
2001
Database
ISI
SICI code
1433-7851(2001)40:21<4040:XCSOAB>2.0.ZU;2-V