Hypervalent iodine in synthesis 81: A one-pot procedure for the synthesis of 1H-imidazole derivatives by cyclocondensation of ketones with [hydroxy(tosyloxy)iodo]benzene and amidines
Pf. Zhang et Zc. Chen, Hypervalent iodine in synthesis 81: A one-pot procedure for the synthesis of 1H-imidazole derivatives by cyclocondensation of ketones with [hydroxy(tosyloxy)iodo]benzene and amidines, SYNTHESIS-S, (14), 2001, pp. 2075-2077
Tosyloxylation of ketones with [hydroxy(tosyloxy)iodo]benzene (HTIB), follo
wed by treatment with amidines provides a one-pot procedure for the synthes
is of 1H-imidazole derivatives with good yields.