A tandem decarboxylation/Diels-Alder reaction of 5-amino-1-phenyl-4-pyrazolecarboxylic acid with 1,3,5-triazines

Authors
Dang, Q Liu, Y Sun, ZL
Citation
Q. Dang et al., A tandem decarboxylation/Diels-Alder reaction of 5-amino-1-phenyl-4-pyrazolecarboxylic acid with 1,3,5-triazines, TETRAHEDR L, 42(48), 2001, pp. 8419-8422
Citations number
22
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
TETRAHEDRON LETTERS
ISSN journal
00404039 → ACNP
Volume
42
Issue
48
Year of publication
2001
Pages
8419 - 8422
Database
ISI
SICI code
0040-4039(20011126)42:48<8419:ATDRO5>2.0.ZU;2-L
Abstract
A tandem decarboxylation/Diels-Alder reaction of 5-amino-1-phenyl-4-pyrazol ecarboxylic acid with various 1,3,5-triazines was reported. The dienophile, 5-amino-1-phenylpyrazole, was generated in situ via decarboxylation and im mediately trapped by 1,3,5-triazines leading to 4,6-disubstituted 1-phenylp yrazolo[3,4-d]pyrimidines in one step. (C) 2001 Elsevier Science Ltd. All r ights reserved.