A combinatorial approach to [1,5]benzothiazepine derivatives as potential antibacterial agents

Authors
Micheli, F Degiorgis, F Feriani, A Paio, A Pozzan, A Zarantonello, P Seneci, P
Citation
F. Micheli et al., A combinatorial approach to [1,5]benzothiazepine derivatives as potential antibacterial agents, J COMB CHEM, 3(2), 2001, pp. 224-228
Citations number
14
Categorie Soggetti
Chemistry & Analysis",Chemistry
Journal title
JOURNAL OF COMBINATORIAL CHEMISTRY
ISSN journal
15204766 → ACNP
Volume
3
Issue
2
Year of publication
2001
Pages
224 - 228
Database
ISI
SICI code
1520-4766(200103/04)3:2<224:ACAT[D>2.0.ZU;2-C
Abstract
[1,5]Benzothiazepines are widely used in a number of different therapeutic areas and therefore represent an interesting scaffold for de novo explorati on. Recent literature reports suggest their value as antibacterial agents. The present paper reports the exploration of this scaffold for the generati on of combinatorial libraries both in solution and on solid phase.