(1S,2S)-2[(S)-Amino(4-methoxyphenyl)methyl]cyclopropan-1-of together with a
range of racemic 2-(2-aminoalkyl)-1-hydroxy-cyclopropanes were prepared by
a stepwise procedure involving a 1,3-dipolar cycloaddition of a nitrile ox
ide to a cyclopropene followed by reduction of the derived bicycle. (C) 200
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