Ma. Brodney et A. Padwa, ELECTROPHILIC AROMATIC-SUBSTITUTION ON PYRIDINE RINGS - INTRAMOLECULAR CYCLIZATION USING N-ACYLIMINIUM IONS, Tetrahedron letters, 38(35), 1997, pp. 6153-6156
The reaction of N-acyliminium ions with several activated pyridines re
sulted in an intramolecular cyclization to provide novel heterocycles.
The reaction exhibited a regiochemical preference for cyclization par
a to the electron donating substitutent. (C) 1997 Elsevier Science Ltd
.