IMPROVED FUNCTIONAL-GROUP COMPATIBILITY IN THE PALLADIUM-CATALYZED AMINATION OF ARYL BROMIDES

Citation
Jp. Wolfe et Sl. Buchwald, IMPROVED FUNCTIONAL-GROUP COMPATIBILITY IN THE PALLADIUM-CATALYZED AMINATION OF ARYL BROMIDES, Tetrahedron letters, 38(36), 1997, pp. 6359-6362
Citations number
13
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
ISSN journal
00404039
Volume
38
Issue
36
Year of publication
1997
Pages
6359 - 6362
Database
ISI
SICI code
0040-4039(1997)38:36<6359:IFCITP>2.0.ZU;2-P
Abstract
Aryl bromides are coupled with amines in the presence of a palladium c atalyst and a stoichiometric amount of cesium carbonate. Using these c onditions base-sensitive functional groups, which were incompatible wi th our previously reported catalytic-amination reaction conditions, ar e well tolerated. (C) 1997 Elsevier Science Ltd.