Jp. Wolfe et Sl. Buchwald, IMPROVED FUNCTIONAL-GROUP COMPATIBILITY IN THE PALLADIUM-CATALYZED AMINATION OF ARYL BROMIDES, Tetrahedron letters, 38(36), 1997, pp. 6359-6362
Aryl bromides are coupled with amines in the presence of a palladium c
atalyst and a stoichiometric amount of cesium carbonate. Using these c
onditions base-sensitive functional groups, which were incompatible wi
th our previously reported catalytic-amination reaction conditions, ar
e well tolerated. (C) 1997 Elsevier Science Ltd.