B. Carboni et al., 1,3-DIPOLAR CYCLOADDITIONS TO UNSATURATED ORGANOBORANES .3. REGIOCONTROLLED AND STEREOCONTROLLED ACCESS TO BORONIC ESTER SUBSTITUTED ISOXAZOLIDINES, Tetrahedron letters, 38(38), 1997, pp. 6665-6668
Alkenylboronic esters undergo regio- and stereoselective 1.3-dipolar c
ycloadditions with nitrones. These reactions give access to boronic es
ter substituted isoxazolidines which can be easily convened by oxidati
on with hydrogen peroxide to the corresponding 4-hydroxy derivatives.
(C) 1997 Elsevier Science Ltd.