AN INVESTIGATION OF THE N-ARYLSULFONYLATION OF 2-AZETIDINONES

Authors
ADLINGTON RM BALDWIN JE MCCOULL W PRITCHARD GJ SCHOFIELD CJ WESTWOOD NJ
Citation
Rm. Adlington et al., AN INVESTIGATION OF THE N-ARYLSULFONYLATION OF 2-AZETIDINONES, Synthetic communications, 27(21), 1997, pp. 3803-3813
Citations number
19
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Synthetic communications → ACNP
ISSN journal
00397911
Volume
27
Issue
21
Year of publication
1997
Pages
3803 - 3813
Database
ISI
SICI code
0039-7911(1997)27:21<3803:AIOTNO>2.0.ZU;2-3
Abstract
N-Arylsulfonylation of 2-azetidinones can lead to the diastereoselecti ve formation of oligomerization products. However, a simple increase o f arylsulfonyl chloride concentration minimized oligomerization and al lowed preparation of 1-arylsulfonyl-2-azetidinones in good yield.