Authors:
TAKEMOTO Y
YUKI H
NISHIDA A
ITO H
KOBAYASHIUCHIDA A
TAKINAMI Y
AKUZAWA S
OHTA M
SATOH M
SEMPLE G
MIYATA K
Citation: Y. Takemoto et al., EFFECTS OF YF476, A POTENT AND SELECTIVE GASTRIN CHOLECYSTOKININ-B RECEPTOR ANTAGONIST, ON GASTRIC-ACID SECRETION IN BEAGLE DOGS WITH GASTRIC FISTULA/, Arzneimittel-Forschung, 48(4), 1998, pp. 403-407
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TAKINAMI Y
YUKI H
NISHIDA A
AKUZAWA S
UCHIDA A
TAKEMOTO Y
OHTA M
SATOH M
SEMPLE G
MIYATA K
Citation: Y. Takinami et al., YF476 IS A NEW POTENT AND SELECTIVE GASTRIN CHOLECYSTOKININ-B RECEPTOR ANTAGONIST IN-VITRO AND IN-VIVO/, Alimentary pharmacology & therapeutics, 11(1), 1997, pp. 113-120
Authors:
YUKI H
NISHIDA A
MIYAKE A
ITO H
AKUZAWA S
TAKINAMI Y
TAKEMOTO Y
MIYATA K
Citation: H. Yuki et al., YM022, A POTENT AND SELECTIVE GASTRIN CCK-B RECEPTOR ANTAGONIST, INHIBITS PEPTONE MEAL-INDUCED GASTRIC-ACID SECRETION IN HEIDENHAIN POUCH DOGS, Digestive diseases and sciences, 42(4), 1997, pp. 707-714
Authors:
SEMPLE G
RYDER H
ROOKER DP
BATT AR
KENDRICK DA
SZELKE M
OHTA M
SATOH M
NISHIDA A
AKUZAWA S
MIYATA K
Citation: G. Semple et al., BENZODIAZEPIN-3-YL)-N'-(3-(METHYLAMINO)PHENYL)UREA (YF476) - A POTENTAND ORALLY-ACTIVE GASTRIN CCK-B ANTAGONIST/, Journal of medicinal chemistry, 40(3), 1997, pp. 331-341
Authors:
SEMPLE G
RYDER H
KENDRICK DA
SZELKE M
OHTA M
SATOH M
NISHIDA A
AKUZAWA S
MIYATA K
Citation: G. Semple et al., SYNTHESIS AND BIOLOGICAL-ACTIVITY OF 1-ALKYLCARBONYLMETHYL ANALOGS OFYM022, Bioorganic & medicinal chemistry letters, 6(1), 1996, pp. 51-54
Authors:
SEMPLE G
RYDER H
KENDRICK DA
SZELKE M
OHTA M
SATOH M
NISHIDA A
AKUZAWA S
MIYATA K
Citation: G. Semple et al., SYNTHESIS AND BIOLOGICAL-ACTIVITY OF 5-HETEROARYL BENZODIAZEPINES - ANALOGS OF YM022, Bioorganic & medicinal chemistry letters, 6(1), 1996, pp. 55-58
Citation: S. Akuzawa et al., [H-3] RAMOSETRON RECOGNIZES 2 BINDING-SITES IN NATIVE AND CLONED RAT 5-HT3 RECEPTORS, The FASEB journal, 10(3), 1996, pp. 807-807
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NISHIDA A
UCHIDAKOBAYASHI A
TAKEMOTO Y
AKUZAWA S
MIYATA K
Citation: A. Nishida et al., COMPARATIVE-EVALUATION OF THE ROLE OF ENDOGENOUS GASTRIN IN BASAL ACID-SECRETION IN CONSCIOUS RATS PROVIDED WITH CHRONIC FISTULA AND PYLORUS LIGATION, Japanese Journal of Pharmacology, 71(3), 1996, pp. 223-230
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KOSHIO H
OHTA M
NISHIDA A
AKUZAWA S
MIYATA K
MASE T
SEMPLE G
Citation: M. Satoh et al., BIOLOGICAL-ACTIVITY OF ANALOGS OF YM022 - NOVEL (3-AMINO SUBSTITUTED PHENYL)UREA DERIVATIVES OF 1,4-BENZODIAZEPIN-2-ONE AS GASTRIN CHOLECYSTOKININ-B RECEPTOR ANTAGONISTS/, Chemical and Pharmaceutical Bulletin, 44(7), 1996, pp. 1412-1414
Citation: S. Akuzawa et al., SELECTIVITY AND THERMAL-PROPERTIES OF VARIOUS STARCHES INCORPORATING FREE FATTY-ACIDS, Bioscience, biotechnology, and biochemistry, 59(9), 1995, pp. 1605-1608
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NISHIDA A
KOBAYASHIUCHIDA A
AKUZAWA S
TAKINAMI Y
SHISHIDO T
KAMATO T
ITO H
YAMANO M
YUKI H
NAGAKURA Y
HONDA K
MIYATA K
Citation: A. Nishida et al., GASTRIN RECEPTOR ANTAGONIST YM022 PREVENTS HYPERSECRETION AFTER LONG-TERM ACID SUPPRESSION, American journal of physiology: Gastrointestinal and liver physiology, 32(5), 1995, pp. 699-705
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ITO H
AKUZAWA S
TSUTSUMI R
KISO T
KAMATO T
NISHIDA A
YAMANO M
MIYATA K
Citation: H. Ito et al., COMPARATIVE-STUDY OF THE AFFINITIES OF THE 5-HT3 RECEPTOR ANTAGONISTS, YM060 YM114 (KAE-393), GRANISETRON AND ONDANSETRON IN RAT VAGUS NERVE AND CEREBRAL-CORTEX, Neuropharmacology, 34(6), 1995, pp. 631-637
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MIYAKE A
MOCHIZUKI S
TAKEMOTO Y
AKUZAWA S
Citation: A. Miyake et al., MOLECULAR-CLONING OF HUMAN 5-HYDROXYTRYPTAMINE(3) RECEPTOR - HETEROGENEITY IN DISTRIBUTION AND FUNCTION AMONG SPECIES, Molecular pharmacology, 48(3), 1995, pp. 407-416
Citation: K. Miyata et al., EFFECT OF SEROTONIN (5-HT)(3)-RECEPTOR ANTAGONISTS YM060, YM114 (KAE-393), ONDANSETRON AND GRANISETRON ON 5-HT4 RECEPTORS AND GASTRIC-EMPTYING IN RODENTS, Japanese Journal of Pharmacology, 69(3), 1995, pp. 205-214
Citation: S. Akuzawa et al., CHARACTERIZATION OF [H-3] YM060, A POTENT AND SELECTIVE 5-HT3 RECEPTOR RADIOLIGAND, IN THE CEREBRAL-CORTEX OF RATS, European journal of pharmacology, 281(1), 1995, pp. 37-42
Authors:
NISHIDA A
TAKINAMI Y
YUKI H
KOBAYASHI A
AKUZAWA S
KAMATO T
ITO H
YAMANO M
NAGAKURA Y
MIYATA K
Citation: A. Nishida et al., YM022 H-1,4-BENZODIAZEPIN-3-YL]-3-(3-METHYLPHENYL)UREA), A POTENT ANDSELECTIVE GASTRIN CHOLECYSTOKININ-B RECEPTOR ANTAGONIST, PREVENTS GASTRIC AND DUODENAL LESIONS IN RATS, The Journal of pharmacology and experimental therapeutics, 270(3), 1994, pp. 1256-1261
Authors:
NISHIDA A
MIYATA K
TSUTSUMI R
YUKI H
AKUZAWA S
KOBAYASHI A
KAMATA T
ITO H
YAMANO M
KATUYAMA Y
SATOH M
OHTA M
HONDA K
Citation: A. Nishida et al., PHARMACOLOGICAL PROFILE OF -1H-1,4-BENZODIAZEPIN-3-YL]-3-(3-METHYLPHENYL)UREA (YM022), A NEW POTENT AND SELECTIVE GASTRIN CHOLECYSTOKININ-BRECEPTOR ANTAGONIST, IN-VITRO AND IN-VIVO, The Journal of pharmacology and experimental therapeutics, 269(2), 1994, pp. 725-731
Authors:
NISHIDA A
TSUTSUMI R
YUKI H
KOBAYASHI A
AKUZAWA S
KAMATO T
ITO H
YAMANO M
MIYATA K
Citation: A. Nishida et al., THE GASTRIN RECEPTOR ANTAGONIST PREVENTS HYPERSECRETORY RESPONSE TO PENTAGASTRIN AFTER LONG-TERM TREATMENT OF OMEPRAZOLE, Gastroenterology, 106(4), 1994, pp. 10000149-10000149
Authors:
YUKI H
NISHIDA A
AKUZAWA S
KOBAYASHI A
TAKINAMI Y
MIYATA K
Citation: H. Yuki et al., GASTRIN PLAYS AN IMPORTANT ROLE ON PEPTONE-INDUCED GASTRIC-ACID SECRETION IN HEIDENHAIN POUCH DOGS, Gastroenterology, 106(4), 1994, pp. 10000215-10000215
Authors:
NISHIDA A
YUKI H
TSUTSUMI R
AKUZAWA S
KOBAYASHI A
TAKINAMI Y
MIYATA K
Citation: A. Nishida et al., YM022, A VERY POTENT AND SELECTIVE GASTRIN CCK-B ANTAGONIST, INHIBITED BASAL AND 2-DEOXY-D-GLUCOSE (2-DG)-INDUCED GASTRIC-ACID SECRETION INRATS, Gastroenterology, 104(4), 1993, pp. 159-159