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Results: 1-15 |
Results: 15
SYNTHESIS AND 5-ALPHA-REDUCTASE INHIBITION-ACTIVITY OF 8-SUBSTITUTED BENZO[F]QUINOLINONES DERIVED FROM PALLADIUM-MEDIATED COUPLING REACTIONS
Authors: SMITH ECR MCQUAID LA GOODE RL MCNULTY AM NEUBAUER BL ROCCO VP AUDIA JE
Citation: Ecr. Smith et al., SYNTHESIS AND 5-ALPHA-REDUCTASE INHIBITION-ACTIVITY OF 8-SUBSTITUTED BENZO[F]QUINOLINONES DERIVED FROM PALLADIUM-MEDIATED COUPLING REACTIONS, Bioorganic & medicinal chemistry letters, 8(4), 1998, pp. 395-398
5-HT1F RECEPTOR AGONISTS INHIBIT NEUROGENIC DURAL INFLAMMATION IN GUINEA-PIGS
Authors: JOHNSON KW SCHAUS JM DURKIN MM AUDIA JE KALDOR SW FLAUGH ME ADHAM N ZGOMBICK JM COHEN ML BRANCHEK TA PHEBUS LA
Citation: Kw. Johnson et al., 5-HT1F RECEPTOR AGONISTS INHIBIT NEUROGENIC DURAL INFLAMMATION IN GUINEA-PIGS, NeuroReport, 8(9-10), 1997, pp. 2237-2240
CHARACTERIZATION OF TYPE-I 5-ALPHA-REDUCTASE ACTIVITY IN DU145 HUMAN PROSTATIC ADENOCARCINOMA CELLS
Authors: KAEFER M AUDIA JE BRUCHOVSKY N GOODE RL HSIAO KC LEIBOVITCH IY KRUSHINSKI JH LEE C STEIDLE CP SUTKOWSKI DM NEUBAUER BL
Citation: M. Kaefer et al., CHARACTERIZATION OF TYPE-I 5-ALPHA-REDUCTASE ACTIVITY IN DU145 HUMAN PROSTATIC ADENOCARCINOMA CELLS, Journal of steroid biochemistry and molecular biology, 58(2), 1996, pp. 195-205
RESPONSES OF LNCAP PROSTATIC ADENOCARCINOMA CELL-CULTURES TO LY300502, A BENZOQUINOLINONE HUMAN TYPE-I 5-ALPHA-REDUCTASE INHIBITOR
Authors: SUTKOWSKI DM AUDIA JE GOODE RL HSIAO KC LEIBOVITCH IY MCNULTY AM NEUBAUER BL
Citation: Dm. Sutkowski et al., RESPONSES OF LNCAP PROSTATIC ADENOCARCINOMA CELL-CULTURES TO LY300502, A BENZOQUINOLINONE HUMAN TYPE-I 5-ALPHA-REDUCTASE INHIBITOR, The Prostate, 1996, pp. 62-66
PICTET-SPENGLER-LIKE SYNTHESIS OF TETRAHYDRO-BETA-CARBOLINES UNDER HYDROLYTIC CONDITIONS - DIRECT USE OF AZALACTONES AS PHENYLACETALDEHYDE EQUIVALENTS
Authors: AUDIA JE DROSTE JJ NISSEN JS MURDOCH GL EVRARD DA
Citation: Je. Audia et al., PICTET-SPENGLER-LIKE SYNTHESIS OF TETRAHYDRO-BETA-CARBOLINES UNDER HYDROLYTIC CONDITIONS - DIRECT USE OF AZALACTONES AS PHENYLACETALDEHYDE EQUIVALENTS, Journal of organic chemistry, 61(22), 1996, pp. 7937-7939
RESOLUTION OF DELTA-LACTAMS PROVIDES ACCESS TO NONRACEMIC BENZOQUINOLINONES - THE SYNTHESIS OF LY300502 AND LY300503
Authors: ASTLEFORD BA AUDIA JE DEETER J HEATH PC JANISSE SK KRESS TJ WEPSIEC JP WEIGEL LO
Citation: Ba. Astleford et al., RESOLUTION OF DELTA-LACTAMS PROVIDES ACCESS TO NONRACEMIC BENZOQUINOLINONES - THE SYNTHESIS OF LY300502 AND LY300503, Journal of organic chemistry, 61(13), 1996, pp. 4450-4454
AMYLOID BETA-MEDIATED OXIDATIVE AND METABOLIC STRESS IN RAT CORTICAL-NEURONS - NO DIRECT EVIDENCE FOR A ROLE FOR H2O2 GENERATION
Authors: ZHANG ZY RYDEL RE DRZEWIECKI GJ FUSON K WRIGHT S WOGULIS M AUDIA JE MAY PC HYSLOP PA
Citation: Zy. Zhang et al., AMYLOID BETA-MEDIATED OXIDATIVE AND METABOLIC STRESS IN RAT CORTICAL-NEURONS - NO DIRECT EVIDENCE FOR A ROLE FOR H2O2 GENERATION, Journal of neurochemistry, 67(4), 1996, pp. 1595-1606
POTENT, SELECTIVE TETRAHYDRO-BETA-CARBOLINE ANTAGONISTS OF THE SEROTONIN 2B (5HT(2B)) CONTRACTILE RECEPTOR IN THE RAT STOMACH FUNDUS
Authors: AUDIA JE EVRARD DA MURDOCH GR DROSTE JJ NISSEN JS SCHENCK KW FLUDZINSKI P LUCAITES VL NELSON DL COHEN ML
Citation: Je. Audia et al., POTENT, SELECTIVE TETRAHYDRO-BETA-CARBOLINE ANTAGONISTS OF THE SEROTONIN 2B (5HT(2B)) CONTRACTILE RECEPTOR IN THE RAT STOMACH FUNDUS, Journal of medicinal chemistry, 39(14), 1996, pp. 2773-2780
COMPARISON OF DESMETHYLSERTRALINE WITH SERTRALINE AS A MONOAMINE UPTAKE INHIBITOR IN-VIVO
Authors: FULLER RW HEMRICKLUECKE SK LITTLEFIELD ES AUDIA JE
Citation: Rw. Fuller et al., COMPARISON OF DESMETHYLSERTRALINE WITH SERTRALINE AS A MONOAMINE UPTAKE INHIBITOR IN-VIVO, Progress in neuro-psychopharmacology & biological psychiatry, 19(1), 1995, pp. 135-149
STEREOSELECTIVE EPOXIDATIONS AND ELECTROPHILIC ADDITIONS TO PARTIAL ERGOT ALKALOIDS AND CONFORMATIONALLY-FIXED STYRENES - EXPERIMENTAL AND THEORETICAL MODELING EVIDENCE FOR THE IMPORTANCE OF TORSIONAL STEERINGAS A STEREOCONTROL ELEMENT
Authors: MARTINELLI MJ PETERSON BC KHAU VV HUTCHISON DR LEANNA MR AUDIA JE DROSTE JJ WU YD HOUK KN
Citation: Mj. Martinelli et al., STEREOSELECTIVE EPOXIDATIONS AND ELECTROPHILIC ADDITIONS TO PARTIAL ERGOT ALKALOIDS AND CONFORMATIONALLY-FIXED STYRENES - EXPERIMENTAL AND THEORETICAL MODELING EVIDENCE FOR THE IMPORTANCE OF TORSIONAL STEERINGAS A STEREOCONTROL ELEMENT, Journal of organic chemistry, 59(8), 1994, pp. 2204-2210
QSAR STUDY OF BENZOQUINOLINONES AS INHIBITORS OF HUMAN TYPE-1 5-ALPHA-REDUCTASE
Authors: WIKEL JH BEMIS KG AUDIA JE MCQUIAD LA JONES CD PENNINGTON PA LAWHORN DE HIRSCH KR STAMM NB
Citation: Jh. Wikel et al., QSAR STUDY OF BENZOQUINOLINONES AS INHIBITORS OF HUMAN TYPE-1 5-ALPHA-REDUCTASE, Bioorganic & medicinal chemistry letters, 3(6), 1993, pp. 1157-1162
SYNTHESIS OF THE INDIVIDUAL ENANTIOMERS OF THE BENZOQUINOLINONE HUMANTYPE-1 STEROID 5-ALPHA-REDUCTASE INHIBITORS LY191704 AND LY266111
Authors: AUDIA JE LAWHORN DE DEETER JB
Citation: Je. Audia et al., SYNTHESIS OF THE INDIVIDUAL ENANTIOMERS OF THE BENZOQUINOLINONE HUMANTYPE-1 STEROID 5-ALPHA-REDUCTASE INHIBITORS LY191704 AND LY266111, Tetrahedron letters, 34(44), 1993, pp. 7001-7004
LY191704 - A SELECTIVE, NONSTEROIDAL INHIBITOR OF HUMAN STEROID 5-ALPHA-REDUCTASE TYPE-1
Authors: HIRSCH KS JONES CD AUDIA JE ANDERSSON S MCQUAID L STAMM NB NEUBAUER BL PENNINGTON P TOOMEY RE RUSSELL DW
Citation: Ks. Hirsch et al., LY191704 - A SELECTIVE, NONSTEROIDAL INHIBITOR OF HUMAN STEROID 5-ALPHA-REDUCTASE TYPE-1, Proceedings of the National Academy of Sciences of the United Statesof America, 90(11), 1993, pp. 5277-5281
SPECIES-DIFFERENCES IN THE PHARMACOLOGY OF THE 5-HYDROXYTRYPTAMINE2 RECEPTOR - STRUCTURALLY SPECIFIC DIFFERENTIATION BY ERGOLINES AND TRYPTAMINES
Authors: NELSON DL LUCAITES VL AUDIA JE NISSEN JS WAINSCOTT DB
Citation: Dl. Nelson et al., SPECIES-DIFFERENCES IN THE PHARMACOLOGY OF THE 5-HYDROXYTRYPTAMINE2 RECEPTOR - STRUCTURALLY SPECIFIC DIFFERENTIATION BY ERGOLINES AND TRYPTAMINES, The Journal of pharmacology and experimental therapeutics, 265(3), 1993, pp. 1272-1279
N(1)-SUBSTITUTED ERGOLINES AND TRYPTAMINES SHOW SPECIES-DIFFERENCES FOR THE AGONIST-LABELED 5-HT(2) RECEPTOR
Authors: JOHNSON MP AUDIA JE NISSEN JS NELSON DL
Citation: Mp. Johnson et al., N(1)-SUBSTITUTED ERGOLINES AND TRYPTAMINES SHOW SPECIES-DIFFERENCES FOR THE AGONIST-LABELED 5-HT(2) RECEPTOR, European journal of pharmacology, 239(1-3), 1993, pp. 111-118
Risultati: 1-15 |