Authors:
Pinto, DJP
Orwat, MJ
Wang, SG
Fevig, JM
Quan, ML
Amparo, E
Cacciola, J
Rossi, KA
Alexander, RS
Smallwood, AM
Luettgen, JM
Liang, L
Aungst, BJ
Wright, MR
Knabb, RM
Wong, PC
Wexler, RR
Lam, PYS
Citation: Djp. Pinto et al., Discovery of 1-[3-(aminomethyl)phenyl]-N-[3-fluoro-2 '- (methylsulfonyl)-[1,1 '-biphenyl]-4-yl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide (DPC423), a highly potent, selective, and orally bioavailable inhibitor of blood coagulation factor Xa, J MED CHEM, 44(4), 2001, pp. 566-578
Authors:
Galemmo, RA
Wells, BL
Rossi, KA
Alexander, RS
Dominguez, C
Maduskuie, TP
Stouten, PFW
Wright, MR
Aungst, BJ
Wong, PC
Knabb, RM
Wexler, RR
Citation: Ra. Galemmo et al., The de novo design and synthesis of cyclic urea inhibitors of factor Xa: Optimization of the S4 ligand, BIOORG MED, 10(3), 2000, pp. 301-304
Citation: J. Cacciola et al., Synthesis and activity studies of conformationally restricted alpha-ketoamide factor Xa inhibitors, BIOORG MED, 10(11), 2000, pp. 1253-1256
Authors:
Han, Q
Dominguez, C
Stouten, PFW
Park, JM
Duffy, DE
Galemmo, RA
Rossi, KA
Alexander, RS
Smallwood, AM
Wong, PC
Wright, MM
Luettgen, JM
Knabb, RM
Wexler, RR
Citation: Q. Han et al., Design, synthesis, and biological evaluation of potent and selective amidino bicyclic factor Xa inhibitors, J MED CHEM, 43(23), 2000, pp. 4398-4415
Authors:
Dominguez, C
Duffy, DE
Han, Q
Alexander, RS
Galemmo, RA
Park, JM
Wong, PC
Amparo, EC
Knabb, RM
Luettgen, J
Wexler, RR
Citation: C. Dominguez et al., Design and synthesis of potent and selective 5,6-fused heterocyclic thrombin inhibitors, BIOORG MED, 9(7), 1999, pp. 925-930
Authors:
Wei, AZ
Smallwood, A
Alexander, RS
Duke, J
Ross, H
Rosenfeld, SA
Chang, CH
Citation: Az. Wei et al., Crystallization and preliminary X-ray diffraction data of the complex of recombinant tick anticoagulant peptide (rTAP) and bovine factor Xa, ACT CRYST D, 55, 1999, pp. 862-864
Authors:
Fevig, JM
Cacciola, J
Alexander, RS
Knabb, RM
Lam, GN
Wong, PC
Wexler, RR
Citation: Jm. Fevig et al., Preparation of meta-amidino-N,N-disubstituted anilines as potent inhibitors of coagulation factor Xa, BIOORG MED, 8(22), 1998, pp. 3143-3148
Citation: Rs. Alexander, No easy walk to freedom: Reconstruction and the ratification of the Fourteenth Amendment., AM J LEG H, 42(2), 1998, pp. 199-200