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Results: 1-10 |
Results: 10
Synthesis of bridged analogs of epibatidine. 3-chloro-5,7,8,9,9a,10-hexahydro-7,10-methanopyrrolo[1,2-b]-2,6-naphthyridine and 2-chloro-5,5a,6,7,8,10-hexahydro-5,8-methanopyrrolo[2,1-b]-1,7-naphthyridine
Authors: Brieaddy, LE Mascarella, SW Navarro, HA Atkinson, RN Damaj, MI Martin, BR Carroll, FI
Citation: Le. Brieaddy et al., Synthesis of bridged analogs of epibatidine. 3-chloro-5,7,8,9,9a,10-hexahydro-7,10-methanopyrrolo[1,2-b]-2,6-naphthyridine and 2-chloro-5,5a,6,7,8,10-hexahydro-5,8-methanopyrrolo[2,1-b]-1,7-naphthyridine, TETRAHEDR L, 42(23), 2001, pp. 3795-3797
Preparation and evaluation of new L-canavanine derivatives as nitric oxidesynthase inhibitors
Authors: Li, XF Atkinson, RN King, SB
Citation: Xf. Li et al., Preparation and evaluation of new L-canavanine derivatives as nitric oxidesynthase inhibitors, TETRAHEDRON, 57(30), 2001, pp. 6557-6565
Factors influencing agonist potency and selectivity for the opioid delta receptor are revealed in structure-activity relationship studies of the 4-[(N-substituted-4-piperidinyl) arylamino]-N,N-diethylbenzamides
Authors: Thomas, JB Herault, XM Rothman, RB Atkinson, RN Burgess, JP Mascarella, SW Dersch, CM Xu, H Flippen-Anderson, JL George, CF Carroll, FI
Citation: Jb. Thomas et al., Factors influencing agonist potency and selectivity for the opioid delta receptor are revealed in structure-activity relationship studies of the 4-[(N-substituted-4-piperidinyl) arylamino]-N,N-diethylbenzamides, J MED CHEM, 44(6), 2001, pp. 972-987
Identification of the first trans-(3R,4R)-dimethyl-4-(3-hydroxyphenyl)piperidine derivative to possess highly potent and selective opioid kappa receptor antagonist activity
Authors: Thomas, JB Atkinson, RN Rothman, RB Fix, SE Mascarella, SW Vinson, NA Xu, H Dersch, CM Lu, YF Cantrell, BE Zimmerman, DM Carroll, FI
Citation: Jb. Thomas et al., Identification of the first trans-(3R,4R)-dimethyl-4-(3-hydroxyphenyl)piperidine derivative to possess highly potent and selective opioid kappa receptor antagonist activity, J MED CHEM, 44(17), 2001, pp. 2687-2690
4-[(8-alkyl-8-azabicyclo[3.2.1]octyl-3-yl)-3-arylanilino]-N,N-diethylbenzamides: High affinity, selective ligands for the delta opioid receptor illustrate factors important to antagonist activity
Authors: Thomas, JB Atkinson, RN Rothman, RB Burgess, JP Mascarella, SW Dersch, CM Xu, H Carroll, FI
Citation: Jb. Thomas et al., 4-[(8-alkyl-8-azabicyclo[3.2.1]octyl-3-yl)-3-arylanilino]-N,N-diethylbenzamides: High affinity, selective ligands for the delta opioid receptor illustrate factors important to antagonist activity, BIOORG MED, 10(11), 2000, pp. 1281-1284
Generation of acyl nitroso compounds by the oxidation of N-acyl hydroxylamines with the Dess-Martin periodinane
Authors: Jenkins, NE Ware, RW Atkinson, RN King, SB
Citation: Ne. Jenkins et al., Generation of acyl nitroso compounds by the oxidation of N-acyl hydroxylamines with the Dess-Martin periodinane, SYN COMMUN, 30(5), 2000, pp. 947-953
Optically pure (-)-4-[(N-allyl-3-methyl-4-piperidinyl)phenyl-amino]-N,N-diethylbenzamide displays selective binding and full agonist activity for thedelta opioid receptor
Authors: Thomas, JB Atkinson, RN Herault, XM Rothman, RB Mascarella, SW Dersch, CM Xu, H Horel, RB Carroll, FI
Citation: Jb. Thomas et al., Optically pure (-)-4-[(N-allyl-3-methyl-4-piperidinyl)phenyl-amino]-N,N-diethylbenzamide displays selective binding and full agonist activity for thedelta opioid receptor, BIOORG MED, 9(23), 1999, pp. 3347-3350
Guanidine-substituted imidazoles as inhibitors of nitric oxide synthase
Authors: Atkinson, RN King, SB
Citation: Rn. Atkinson et Sb. King, Guanidine-substituted imidazoles as inhibitors of nitric oxide synthase, BIOORG MED, 9(20), 1999, pp. 2953-2958
Asymmetric synthesis of conformationally restricted L-arginine analogues as active site probes of nitric oxide synthase
Authors: Atkinson, RN Moore, L Tobin, J King, SB
Citation: Rn. Atkinson et al., Asymmetric synthesis of conformationally restricted L-arginine analogues as active site probes of nitric oxide synthase, J ORG CHEM, 64(10), 1999, pp. 3467-3475
Synthesis and evaluation of new sulfur-containing L-arginine-derived inhibitors of nitric oxide synthase
Authors: Ichimori, K Stuehr, DJ Atkinson, RN King, SB
Citation: K. Ichimori et al., Synthesis and evaluation of new sulfur-containing L-arginine-derived inhibitors of nitric oxide synthase, J MED CHEM, 42(10), 1999, pp. 1842-1848
Risultati: 1-10 |